平安! 发表于 2011-11-9 19:57
2 D. _8 r* J8 Z$ ^3 ePazopanib (100 mg/kg/day free base equivalent)
1 ^, I. V& Z) o) G+ n$ `6 E 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。/ O, O& n: @& N
搜索了一下,原料一大堆。( Y: M: \ v2 U" f+ A' A: q
7 Q, V8 w) c/ v) @% q7 |7 x* M对不起!100mg/kg是用于移植瘤的,我弄错了。* K) D1 ~4 t7 y, Z& l2 R8 J5 \1 |
, }7 v/ T0 i% E0 e6 ^; ^以下是正版说明书的推荐用量。$ f: V" h$ v, T% E( v: j/ [& W2 ^3 E
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--------------------- DOSAGE AND ADMINISTRATION ----------------3 N$ ^5 h6 V6 n. ?5 V
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) / A; @3 O9 Q/ I
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) 8 V% l/ O5 G0 H" i) M r E
---------------------DOSAGE FORMS AND STRENGTHS --------------" n1 A. M% g: E/ Q j, o0 @
200 mg tablets. (3) & }/ S3 W- ]/ N
-------------------------------CONTRAINDICATIONS------------------------ |